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The Pharmaceutical Society of Korea (대한약학회)
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A Convergent Synthetic Study of Biologically Active Benzofuran Derivatives

  • Hu, Kun (College of Pharmacy, Kyung Hee University) ;
  • Jeong, Jin-Hyun (College of Pharmacy, Kyung Hee University)
  • Published : 2006.06.01
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Abstract

In order to construct a benzofuran library, we developed a model study of benzbromarone. Synthesis has been achieved in 53% overall yield, starting from phenol via the key intermediate 2-ethylbenzofuran which was afforded by intramolecular Wittig reaction.

Keywords

References

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