References
- Daluge, S. M., Good, S. S., Faletto, M. B., Miller, W. H., St Clair, M. H., Boone, L. R., Tisdale, M., Parry, N. R., Reardon, J. E., Dornsife, R. E., Averett, D. R., and Krenitsky, T. A., A novel carbocyclic nucleoside analog with potent, selective antihuman immunodeficiency virus activity. Antimicrob. Agents Chemother., 41, 1082-1093 (1997)
-
Furman, P. A., Fyfe, J. A., St. Clair, M. H., Weinhold, K., Rideout, J. L., Freeman, G. A., Nusinoff-Lehrman, S., Bolognesi, D. P., Broder, S., Mitsuya, H., and Barry, D. W., Phosphorylation of 3
$¢$ -azido-3$¢$ -deoxythymidine and selective interaction of the 5¢-triphosphate with human immunodeficiency virus reverse transcriptase. Proc. Natl. Acad. Sci. U.S.A., 83, 8333-8337 (1986) -
Hong, J. H. and Ok, O. H., Synthesis of 4'-
${\alpha}$ -C phenyl-branched carbocyclic nucleoside using ring-closing metathesis. Bull. Korean Chem. Soc., 24, 1289-1292 (2003) https://doi.org/10.5012/bkcs.2003.24.9.1289 - Lin, T.-S., Schinazi, R. F., and Prusoff, W. H., Potent and selective in vitro activity of 3'-deoxy thymidine-2'-ene (3'- deoxy-2',3'-dideoxydehydrothymidine) against human immunodeficiency virus. Biochem. Pharmacol., 36, 2713-2718 (1987) https://doi.org/10.1016/0006-2952(87)90253-X
- Nair, V. and Tahnke, T., Antiviral activities of isomeric dideoxynucleosides of D- and L-related stereochemistry. Antimicrob. Agents Chemother., 39, 1017-1029 (1995) https://doi.org/10.1128/AAC.39.5.1017
- Nair, V., Zintek, L. B., Sells, T. B., Jeffery, A. L., Nuesca, Z. M., Purdy, D. F., Jeon, G. S., Hamilton, R. B., Bolon, P. J., and Malany, S., Novel chiral isomeric nucleosides and nucleotides: Synthesis, enzymology, and anti-HIV activity. Antiviral Res., 23, 38-38 (1994)
-
Ohrui, H., Kohgo, S., Kitano, K., Sakata, S., Kodama, E., Yoshimura, K., Matsuoka, M., Shigeta, S., and Mitsuya, H., Synthesis of 4'-C-ethynyl-
${\beta}$ -D-arabino- and 4'-C-ethynyl-2'- deoxy-${\beta}$ -D-ribo-pentofuranosylpyrimidines and -purines and evaluation of their anti-HIV activity. J. Med. Chem., 43, 4516- 4525 (2000) https://doi.org/10.1021/jm000209n - O-Yang, C., Wu, H. Y., Fraser-Smith, E. B., and Walker, K. A. M., Synthesis of 4'-cyanothymidine and analogs as potent inhibitors of HIV. Tetrahedron Lett., 33, 37-40 (1992) https://doi.org/10.1016/S0040-4039(00)77667-2
- Schinazi, R. F., Chu, C. K., Peck, A., McMillan, A., Mathis, R., Cannon, D., Jeong, L. S., Beach, J. W., Choi, W. B., Yeola, S., and Liotta, D. C., Activities of the four optical isomers of 2',3'-dideoxy-3'-thiacytidine (BCH-189) against human immunodeficiency virus type I in human lymphocytes. Antimicrob. Agents Chemother., 36, 672-676 (1992) https://doi.org/10.1128/AAC.36.3.672
- Sells, T. B. and Nair, V., Synthetic approaches to novel isomeric dideoxynucleosides containing a chiral furanethanol carbohydrate moiety. Tetrahedron Lett., 34, 3527-3530 (1993) https://doi.org/10.1016/S0040-4039(00)73627-6
-
Sugimoto, I., Shuto, S., Mori, S., Shigeta, S., Matuda, A., Synthesis of 4'
${\alpha}$ -branched thymidines as a new type of antiviral agents. Bioorg. Med. Chem. Lett., 9, 385-388 (1999) https://doi.org/10.1016/S0960-894X(99)00010-4 - Yarchoan, R., Mitsuya, H., Thomas, R. V., Pluda, J. M., Hartman, N. R., Perno, C. F., Marczyk, K. S., Allain, J.-P., Johns, D. G., and Broder, S., In vivo activity against HIV and favorable toxicity profile of 2',3'-dideoxyinosine. Science, 245, 412-415 (1989) https://doi.org/10.1126/science.2502840
- Yarchoan, R., Thomas, R. V., Allain, J.-P., McAtee, N., Dubinsky, R., Mitsuya, H., Lawley, T. J., Safai, B., Myers, C. E., Perno, C. F., Klecker, R. W., Wills, R. J., Fischl, M. A., McNeely, M. C., Pluda, J. M., Leuther, M., Collins, J. M., and Broder, S. The phase I studies of 2',3'-dideoxycytidine in human immunodeficiency virus infection as single agent and alternating with zidovudine (AZT). Lancet ,1, 76-81 (1988)