DOI QR코드

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Biological Evaluation and Molecular Docking Study of 3-(4-Sulfamoylphenyl)-4-phenyl-1H-pyrrole-2,5-dione as COX-2 Inhibitor

  • Pham, Van Chung (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Shin, Ji-Sun (Department of Pharmaceutical Biochemistry and Department of Life and Nanopharmaceutical Science, College of Pharmacy, Kyung Hee University) ;
  • Choi, Min-Ji (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Kim, Tae-Woo (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Lee, Ki-Jae (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Kim, Kyung-Ju (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Huh, Geun (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Kim, Jung-Ahn (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Choo, Dong-Joon (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Lee, Kyung-Tae (Department of Pharmaceutical Biochemistry and Department of Life and Nanopharmaceutical Science, College of Pharmacy, Kyung Hee University) ;
  • Lee, Jae-Yeol (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
  • 투고 : 2011.09.14
  • 심사 : 2011.12.14
  • 발행 : 2012.02.20

초록

키워드

참고문헌

  1. Chandrasekharan, N. V.; Dai, H.; Roos, K. L.; Evanson, N. K.; Tomsik, J.; Elton, T. S.; Simmons, D. L. Proc. Natl. Acad. Sci. U.S.A. 2002, 99, 13926. https://doi.org/10.1073/pnas.162468699
  2. Lee, S. H.; Kim, M. H.; Han, H. J. Am. J. Physiol. Cell Physiol. 2009, 297, C207. https://doi.org/10.1152/ajpcell.00579.2008
  3. Watson, D. J.; Harper, S. E.; Zhao, P.-L.; Quan, H.; Bolognese, J. A.; Simon, T. J. Arch. Intern. Med. 2000, 160, 2998. https://doi.org/10.1001/archinte.160.19.2998
  4. Hawkey, C. J. Lancet 1999, 353, 307. https://doi.org/10.1016/S0140-6736(98)12154-2
  5. Chan, F. K.; Hung, L. C.; Suen, B. Y.; Wu, J. C.; Lee, K. C.; Leung, V. K.; Hui, A. J.; To, K. F.; Leung, W. K.; Wong, V. W.; Chung, S. C.; Sung, J. J. N. Engl. J. Med. 2002, 347, 2104. https://doi.org/10.1056/NEJMoa021907
  6. McGettigan, P.; Henry, D. JAMA 2006, 296, 1633. https://doi.org/10.1001/jama.296.13.jrv60011
  7. Mason, R. P.; Walter, M. F.; McNulty, H. P.; Lockwood, S. F.; Byun, J.; Day, C. A.; Jacob, R. F. J. Cardiovasc. Pharmacol. 2006, 47, S7. https://doi.org/10.1097/00005344-200605001-00003
  8. Moon, J. T.; Jeon, J. Y.; Park, H. A.; Noh, Y. S.; Lee, K. T.; Kim, J.; Choo, D. J.; Lee, J. Y. Bioorg. Med. Chem. Lett. 2010, 20, 734. https://doi.org/10.1016/j.bmcl.2009.11.067
  9. Yun, K. J.; Shin, J. S.; Choi, J. H.; Back, N. I.; Chung, H. G.; Lee, K. T. Int. Immunopharmacol. 2009, 9, 1323. https://doi.org/10.1016/j.intimp.2009.08.001
  10. Uddin, M. J.; Praveen Rao, P. N.; Knaus, E. E. Bioorg. Med. Chem. 2004, 12, 5929. https://doi.org/10.1016/j.bmc.2004.08.021
  11. Churchill, L.; Graham, A. G.; Shih, C.-K.; Pauletti, D.; Farina, P. R.; Grob, P. M. Inflammopharmacology 1996, 4, 125. https://doi.org/10.1007/BF02735467
  12. Manivannan, E.; Chaturvedi, S. C. Bioorg. Med. Chem. 2011, 19,4520. https://doi.org/10.1016/j.bmc.2011.06.019
  13. Abdel-Aziz, A. A.; ElTahir, K. E.; Asiri, Y. A. Eur. J. Med. Chem. 2011, 46, 1648. https://doi.org/10.1016/j.ejmech.2011.02.013
  14. Gautam, R.; Jachak, S. M.; Kumar, V.; Mohan, C. G. Bioorg. Med. Chem. Lett. 2011, 21, 1612. https://doi.org/10.1016/j.bmcl.2011.01.116
  15. Singh, P.; Bhardwaj, A.; Kaur, S.; Kumar, S. Eur. J. Med. Chem. 2009, 44, 1278. https://doi.org/10.1016/j.ejmech.2008.08.008
  16. MVD 2010.4.2 for Windows in Molegro ApS.
  17. Selinsky, B. S.; Gupta, K.; Sharkey, C. T.; Loll, P. J. Biochemistry 2001, 40, 5172. https://doi.org/10.1021/bi010045s
  18. Wang, J. L; Limburg, D.; Graneto, M. J.; Springer, J.; Hamper, J. R.; Liao, S.; Pawlitz, J. L.; Kurumbail, R. G.; Maziasz. T.; Talley, J. J.; Kiefer, J. R.; Carter, J. Bioorg. Med. Chem. Lett. 2010, 20, 7159. https://doi.org/10.1016/j.bmcl.2010.07.054

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  2. Synthesis of Pyrroles and Condensed Pyrroles as Anti-Inflammatory Agents with Multiple Activities and Their Molecular Docking Study vol.05, pp.04, 2015, https://doi.org/10.4236/ojmc.2015.54005
  3. Ultrasonic synthesis, characterization, and antibacterial evaluation of novel heterocycles containing hexahydroquinoline and pyrrole moieties vol.23, pp.1, 2012, https://doi.org/10.1515/hc-2016-0164
  4. Ultrasonic synthesis, characterization, and antibacterial evaluation of novel heterocycles containing hexahydroquinoline and pyrrole moieties vol.23, pp.1, 2012, https://doi.org/10.1515/hc-2016-0164