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Exploration of Novel Ureidobenzothiazole Library Against Neuroinflammation

  • Han, Min-Soo (Organic Chemistry Laboratory, Korea Institute of Science and Technology) ;
  • Park, Chan-Ho (Organic Chemistry Laboratory, Korea Institute of Science and Technology) ;
  • Nam, Kee-Dal (Organic Chemistry Laboratory, Korea Institute of Science and Technology) ;
  • Cho, Sung-Woo (Department of Biochemistry and Molecular Biology, University of Ulsan college of Medicine) ;
  • Hahn, Hoh-Gyu (Organic Chemistry Laboratory, Korea Institute of Science and Technology)
  • Received : 2011.07.08
  • Accepted : 2011.08.23
  • Published : 2011.10.20

Abstract

Keywords

References

  1. Muller, G. Drug Discov. Today 2003, 8, 681-691. https://doi.org/10.1016/S1359-6446(03)02781-8
  2. Bonne, C.; Muller, A.; Latour, E.; Tissie, G.; Emerit, I.; Modat, G.; Dornand, J.; Roch, M.; Giroud, J. P.; Griswold, D. E.; Marshall, P. J.; Coquelet, C. Arzneimittelforschung 1989, 39, 1242-1245.
  3. Rickles, R.; Lee, M. S. PCT Int. Appl. WO 2009011893, 2009; p 70.
  4. Rickles, R.; Pierce, L.; Lee, M. S. PCT Int. Appl. WO 2009011897, 2009; p 79.
  5. Andersen, C. B.; Wan, Y.; Chang, J. W.; Riggs, B.; Lee, C.; Liu, Y.; Sessa, F.; Villa, F.; Kwiatkowski, N.; Suzuki, M.; Nallan, L.; Heald, R.; Musacchio, A.; Gray, N. S. ACS Chemical Biology 2008, 3, 180-192. https://doi.org/10.1021/cb700200w
  6. Helal, C. J.; Sanner, M. A.; Cooper, C. B.; Gant, T.; Adam, M.; Lucas, J. C.; Kang, Z.; Kupchinsky, S.; Ahlijanian, M. K.; Tate, B.; Menniti, F. S.; Kelly, K.; Peterson, M. Bioorg. Med. Chem. Lett. 2004, 14, 5521-5525. https://doi.org/10.1016/j.bmcl.2004.09.006
  7. Shimamura, T.; Shibata, J.; Kurihara, H.; Mita, T.; Otsuki, S.; Sagara, T.; Hirai, H.; Iwasawa, Y. Bioorg. Med. Chem. Lett. 2006, 16, 3751-3754. https://doi.org/10.1016/j.bmcl.2006.04.048
  8. Subramanian, R.; Lee, M. R.; Allen, J. G.; Bourbeau, M. P.; Fotsch, C.; Hong, F.-T.; Tadesse, S.; Yao, G.; Yuan, C. C.; Surapaneni, S.; Skiles, G. L.; Wang, X.; Wohlhieter, G. E.; Zeng, Q.; Zhou, Y.; Zhu, X.; Li, C. Chem. Res. Toxicol. 2010, 23, 653- 663. https://doi.org/10.1021/tx900414g
  9. Das, J.; Chen, P.; Norris, D.; Padmanabha, R.; Lin, J.; Moquin, R. V.; Shen, Z.; Cook, L. S.; Doweyko, A. M.; Pitt, S.; Pang, S.; Shen, D. R.; Fang, Q.; de Fex, H. F.; McIntyre, K. W.; Shuster, D. J.; Gillooly, K. M.; Behnia, K.; Schieven, G. L.; Wityak, J.; Barrish, J. C. J. Med. Chem. 2006, 49, 6819-6832. https://doi.org/10.1021/jm060727j
  10. Suzuki, H.; Hibi, T. Neurogastroenterol. Motil. 2010, 22, 595- 599. https://doi.org/10.1111/j.1365-2982.2010.01486.x
  11. Tack, J.; Masclee, A.; Heading, R.; Berstad, A.; Piessevaux, H.; Popiela, T.; Vandenberghe, A.; Kato, H. Neurogastroenterol. Motil. 2009, 21, 272-280. https://doi.org/10.1111/j.1365-2982.2009.01261.x
  12. Matsueda, K.; Hongo, M.; Tack, J.; Aoki, A.; Saito, Y.; Kato, H. Neurogastroenterol. Motil. 2010, 22, 618-e173. https://doi.org/10.1111/j.1365-2982.2009.01449.x
  13. Gallardo-Godoy, A.; Gever, J.; Fife, K. L.; Silber, B. M.; Prusiner, S. B.; Renslo, A. R. J. Med. Chem. 2011, 54, 1010-1021. https://doi.org/10.1021/jm101250y
  14. Bolognesi, M. L.; Bartolini, M.; Tarozzi, A.; Morroni, F.; Lizzi, F.; Milelli, A.; Minarini, A.; Rosini, M.; Hrelia, P.; Androsano, V.; Melchiorre, C. Bioorg. Med. Chem. Lett. 2011, 21, 2655-2658. https://doi.org/10.1016/j.bmcl.2010.12.093
  15. Choi, M.-M.; Kim, E.-A.; Hahn, H.-G.; Nam, K. D.; Yang, S.-J.; Choi, S. Y.; Kim, T. U.; Cho, S.-W.; Huh, J.-W. Toxicology 2007, 239, 156-166. https://doi.org/10.1016/j.tox.2007.07.010
  16. Katritzky, A. R.; Tymoshenko, D. O.; Monteux, D.; Vvedensky, V.; Nikonov, G.; Cooper, C. B.; Deshpande, M. J. Org. Chem. 2000, 65, 8059-8062. https://doi.org/10.1021/jo000946r
  17. Cody, R. B.; Laramée, J. A.; Durst, H. D. Anal. Chem. 2005, 77, 2297-2302. https://doi.org/10.1021/ac050162j
  18. Kim, E.-A.; Hahn, H.-G.; Kim, K.-S.; Kim, T. U.; Choi, S. Y.; Cho, S.-W. Cell. Mol. Neurobiol. 2010, 30, 807-815. https://doi.org/10.1007/s10571-010-9508-x
  19. Kim, E.- A.; Kim, H.; Ahn, J.-Y.; Hahn, H.-G.; Kim, K.-S.; Kim, T. U.; Cho, S.-W. Mol. Cells 2010, 30, 51-57. https://doi.org/10.1007/s10059-010-0087-y