Barbiturates as Noncompetitive Inhibitors of PTP1B and Competitive Inhibitors of Vaccinia H1-Related (VHR) Phosphatase

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Khadka, Deegendra (Department of Chemistry, College of Natural Sciences, Inha University) ;
Kafle, Bhooshan (Department of Chemistry, College of Natural Sciences, Inha University) ;
Park, Hwang-Seo (Department of Bioscience and Biotechnology, College of Engineering, Sejong University) ;
Cho, Hyeong-Jin (Department of Chemistry, College of Natural Sciences, Inha University)

Ho, I. K.; Harris, R. A. Ann. Rev. Pharmacol. Toxicol. 1981, 21, 83. https://doi.org/10.1146/annurev.pa.21.040181.000503
Rosenfeld, G. C., Loose, D. S., Eds.; Pharmacology, 3rd ed.; Lippincott Williams & Wilkins: Baltimore, 2007; pp 101-147.
Kafle, B.; Bhattarai, B. R.; Cho, H. Bull. Korean Chem. Soc. 2011, 32, 31 https://doi.org/10.5012/bkcs.2011.32.1.31
Humar, M.; Pischke, S. E.; Loop, T.; Hoetzel, A.; Schmidt, R.; Klaas, C.; Pahl, H. L.; Geiger, K. K.; Pannen, B. H. J. Mol. Pharmacol. 2004, 65, 350. https://doi.org/10.1124/mol.65.2.350
Park, H.; Bhattarai, B. B.; Ham, S. W.; Cho, H. Eur. J. Med. Chem. 2009, 44, 3280. https://doi.org/10.1016/j.ejmech.2009.02.011
Bruckmann, G.; Isaacs, S. D. J. Am. Chem. Soc. 1949, 71, 390. https://doi.org/10.1021/ja01170a004
Laudien, R.; Mitzner, R. J. Chem. Soc., Perkin Trans. 2001, 2, 2226.
Can. J. Chem. 1981, 59, 2629 https://doi.org/10.1139/v81-379
Tetrahedron Lett. 1995, 36, 3103 https://doi.org/10.1016/0040-4039(95)00478-U
Santoso, M. J. Mat. & Sains 2000, 5, 91.
Yuvaniyama, J.; Denu, J. M.; Dixon, J. E.; Saper, M. A. Science 1996, 272, 1328. https://doi.org/10.1126/science.272.5266.1328

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