References
- De Souza, E. M., Menna-Barreto, R., Araujo-Jorge, T. C., Kumar, A., Hu, Q., Boykin, D. W. and Soeiro, M. N. C. (2006) Antiparasitic activity of aromatic diamidines is related to apoptosis-like death in Trypanosoma cruzi. Parasitology 133, 75-79. https://doi.org/10.1017/S0031182006000084
- Bailly, C., Perrine, D., Lancelot, J. C., Saturnino, C., Robba, M. and Waring, M. J. (1997) Sequence-selective binding to DNA of bis (amidinophenoxy) alkanes related to propamidine and pentamidine. Biochem. J. 323, 23-31. https://doi.org/10.1042/bj3230023
- Tabernero, L., Bella, J. and Aleman, C. (1996) Hydrogen bond geometry in DNA-minor groove binding drug complexes. Nucleic. Acids Res. 24, 3458-3466. https://doi.org/10.1093/nar/24.17.3458
- Nguyen, B., Lee, M. P. H., Iberg, D. H., Joubert, A., Bailly, C., Brun, R., Neidle, S. and Wilson, W. D. (2002) Strong binding in the DNA minor groove by an aromatic diamidine with a shape that does not match the curvature of the groove. JACS. 124, 13680-13681. https://doi.org/10.1021/ja027953c
- Lansiaux, A., Tanious, F., Mishal, Z., Dassonneville, L., Kumar, A., Stephens, C. E., Hu, Q., Wilson, W. D., Boykin, D. W. and Bailly, C. (2002) Distribution of furamidine analogues in tumor cells: targeting of the nucleus or mitochondria depending on the amidine substitution. Cancer Res. 62, 7219-7229.
- Miletti, K. E. and Leibowitz, M. J. (2000) Pentamidine inhibition of group I intron splicing in Candida albicans correlates with growth inhibition. Antimicrob. Agents Chemother. 44, 958-966. https://doi.org/10.1128/AAC.44.4.958-966.2000
- Zhang, Y., Li, Z. J., Pilch, D. S. and Leibowitz. M. J. (2002) Pentamidine inhibits catalytic activity of group I intron Ca.LSU by altering RNA folding. Nucleic. Acids Res. 30, 2961-2971. https://doi.org/10.1093/nar/gkf394
- Bielawski, K., Galicka, A., Bielawska, A. and Sredzinska, K. (2000) Inhibitory effects of pentamidine analogues on protein biosynthesis in vitro. Acta. Biochimica. Polonica. 47, 113-120.
- Lanteri, C. A., Trumpower, B. L., Tidwell, R. R. and Meshnick, S. R. (2004) DB75, a novel trypanocidal agent, disrupts mitochondrial function in Saccharomyces cerevisiae. Antimicrob. Agents Chemother. 48, 3968-3974. https://doi.org/10.1128/AAC.48.10.3968-3974.2004
- Werbovetz, K. (2006) Diamidines as antitrypanosomal, antileishmanial and antimalarial agents. Curr. Opin. Investig. Drugs 7, 147-157.
- Mathis, A. M., Holman, J. L., Sturk, L. M., Ismail, M. A., Boykin, D. W., Tidwell, R. R. and Hall, J. E. (2006) Accumulation and intracellular distribution of antitrypanosomal diamidine compounds DB75 and DB820 in African trypanosomes. Antimicrob. Agents Chemother. 50, 2185-2191. https://doi.org/10.1128/AAC.00192-06
- Montgomery, A. B., Debs, R. J., Luce, J. M., Corkery, K. J., Turner, J., Brunette, E. N., Lin, E. T. and Hopewell, P. C. (1987) Aerosolised pentamidine as sole therapy for Pneumocystis carinii pneumonia in patients with acquired immunodeficiency syndrome. Lancet II 2, 480-483.
- Lanteri, C. A., Stewart, M. L., Brock, J. M., Alibu, V. P., Meshnick, S. R., Tidwell, R. R. and Barrett, M. P. (2006) Roles for the Trypanosoma brucei P2 transporter in DB75 uptake and resistance. Mol. Pharmacol. 70, 1585-1592. https://doi.org/10.1124/mol.106.024653
- Lourie, E. M. and Yorke, W. (1939) The trypanocidal action of certain aromatic diamidines. Ann. Trop. Med. Para. 33, 289-304. https://doi.org/10.1080/00034983.1939.11685073
- Elson., W. O. (1945) The antibacterial and fungistatic properties of propamidine. J. Infect. Dis. 76, 193-197. https://doi.org/10.1093/infdis/76.3.193
- Chen, A. L., He, J., Lian, Y. J., Feng, J. T. and Zhang, X. (2006) The fungicide activity of analogs of pentamidine against Botrytis cinerea. J. Plant Protection 33, 68-72.
- Wu, W. J. (1987) Experiment technology of plant chemical protection. Shaanxi Science and Technology Press, Xi’an, China.
- Walzer, P. D., Kim, C. K., Foy, J., Linke, M. J. and Cushion, M. T. (1988) Cationic antitrypanosomal and other antimicrobial agents in the therapy of experimental Pneumocystis carinii pneumonia. Antimicrob. Agents Chemother. 32, 896-905. https://doi.org/10.1128/AAC.32.6.896
- Gazzard, B. G. (1989) Pneumocystis carinii pneumonia and its treatment in patients with AIDS. J. Antimicrob. Chemother. 23, 67-75. https://doi.org/10.1093/jac/23.suppl_A.67
- Wispelwey, B. and Pearson, R. D. (1991) Pentamidine: a review, In-fect. Infect. Control Hosp. Epidemiol. 12, 375-381. https://doi.org/10.1086/646360
- Varga, J. H., Wolf, T. C., Jensen, H. G., Parmley, V. C. and Rowsey, J. J. (1993) Combined treatment of Acanthamoeba keratitis with propamidine, neomycin, and polyhexamethylene biguanide. Am. J. Ophthalmol. 115, 466-470. https://doi.org/10.1016/S0002-9394(14)74448-4
- Perrine, D., Chenu, J. P., Georges, P., Lancelot, J. C., Saturnino, C. and Robba. M. (1995) Effect of zidovudine on transplacental pharmacokinetics of ddI in the pigtailed macaque (Macaca nemestrina). Antimicrob. Agents Chemother. 39, 339-342. https://doi.org/10.1128/AAC.39.2.339
- Chen, A. L., He, J., Lian, Y. J., Feng, J. T. and Zhang, X. (2006) The fungicide activity of analogs of pentamidine against Botrytis cinerea. Acta. Phytophylacica Sinica. 33, 68-72.
- Luck, G., Zimmer, C. and Schweizer, D. (1988) DNA binding studies of the nonintercalative ligand pentamidine: dA-dT basepair preference. Studia Biophys. 125, 107-119.
- Fox, K. R., Sansom, C. E. and Stevens, M. F. G. (1990) Footprinting studies on the sequence-selective binding of pentamidine to DNA. FEBS Letters 266, 150-154. https://doi.org/10.1016/0014-5793(90)81527-U
- Lanteri, C. A., Tidwell, R. R. and Meshnick, S. R. (2008) The mitochondrion is a site of trypanocidal action of the aromatic diamidine DB75 in bloodstream forms of Trypanosoma brucei. Antimicrob. Agents Chemother. 52, 875-882. https://doi.org/10.1128/AAC.00642-07
- Kang, Z. (1996) Ultrastructure of Plant Pathogenic Fungi, Chain Science and Technology Press, Beijing.
- Yoneyama, K. and Misato, T. (1971) Studies on the fungicidal action of dithiocarbamates. Ann. Phytopath. Soc. Japan 37, 291-300. https://doi.org/10.3186/jjphytopath.37.291
- Chance, B. and Willium, G. R. (1955) Respiration enzymes in oxidative phosphorylation. I. Kinetics of oxygen utilization. J. Biol. Chem. 217, 383-393.
- Pecci, L., Montefoschi, G., Fontana, M. and Cavallini, D. (1994) Aminoethylcysteine ketimine decarboxylated dimer inhibits mitochondrial respiration by impairing electron transport at complex I level. Biochem. Biophys. Res. Commun. 199, 755-760. https://doi.org/10.1006/bbrc.1994.1293
- Singer, T. P. (1974) Determination of the activity of succinate, NADH, choline, and alpha-glycerophosphate dehydrogenases. Methods Biochem. Anal. 22, 123-175. https://doi.org/10.1002/9780470110423.ch3
- Hatefi, Y. and Stiggall, D. L. (1978) Preparation and properties of succinate: ubiquinonereductase (ComplexII). Methods Enzymol. 53, 21-27. https://doi.org/10.1016/S0076-6879(78)53008-5
- Krahenbuhl, S., Chang, M., Brass, E. P. and Hoppel, C. L. (1991) Decreased activities of ubiquinol: ferricytochrome c oxidoreductase (complex III) and ferrocytochromec: oxygen oxidoreductase (complex IV) in liver mitochondria from rats with hydroxycobalamin (c-lactam)-induced methylmalonic aciduria. J. Biol. Chem. 266, 20998-21003.
- Boffoli, D., Scacco, S. C., Vergari, R., Solarin, G., Santacroce, G. and Papa, S. (1994) Decline with age of the respiratory chain activity in human skeletal muscle. Biochim. Biophys. Acta. 1226, 73-82. https://doi.org/10.1016/0925-4439(94)90061-2
Cited by
- Therapeutic agents and biocides for ocular infections by free-living amoebae of Acanthamoeba genus vol.62, pp.2, 2017, https://doi.org/10.1016/j.survophthal.2016.10.009
- Diamidine Compounds for Selective Inhibition of Protein Arginine Methyltransferase 1 vol.57, pp.6, 2014, https://doi.org/10.1021/jm401884z