Bulletin of the Korean Chemical Society

Korean Chemical Society (대한화학회)
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Synthesis and Biological Evaluation of 2-Aminoisonicotinic Acid Analogues as HIF-1α Inhibitors

  • Received : 2010.09.02
  • Accepted : 2010.09.27
  • Published : 2010.12.20
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Abstract

Keywords

References

  1. Jiang, B. H.; Rue, E.; Wang, G. L.; Roe, R.; Semenza, G. L. J. Biol. Chem. 1996, 2711, 7771-17778.
  2. Wang, G. L.; Semenza, G. L. J. Biol. Chem. 1995, 270, 1230-1237. https://doi.org/10.1074/jbc.270.3.1230
  3. Semenza, G. L. Nat. Rev. Cancer 2003, 3, 721-732. https://doi.org/10.1038/nrc1187
  4. Pili, R.; Donehower, R. C. J. Natl. Cancer Inst. 2003, 95, 498-499. https://doi.org/10.1093/jnci/95.7.498
  5. Shin, D. H.; Kim, J. H.; Jung, Y. J.; Kim, K. E.; Jeong, J. M.; Chun, Y. S.; Park, J. W. Cancer Lett. 2007, 255, 107-116. https://doi.org/10.1016/j.canlet.2007.03.026
  6. Dikmen, Z. G.; Gellert, G. C.; Dogan, P.; Yoon, H.; Lee, Y. B.;Ahn, C. H.; Shay, J. W. J. Cell Biochem. 2008, 104, 985-994. https://doi.org/10.1002/jcb.21681
  7. Cai, X. F.; Jin, X.; Lee, D.; Yang, Y. T.; Lee, K.; Hong, Y. S.; Lee,J. H.; Lee, J. J. J. Nat. Prod. 2006, 69, 1095-1097. https://doi.org/10.1021/np060081y
  8. Lee, K.; Lee, J. H.; Boovanahalli, S. K.; Jin, Y.; Lee, M.; Jin, X.;Kim, J. H.; Hong, Y. S.; Lee, J. J. J. Med. Chem. 2007, 50, 1675-1684. https://doi.org/10.1021/jm0610292
  9. Boovanahalli, S. K.; Jin, X.; Jin, Y.; Kim, J. H.; Dat, N. T.; Hong,Y. S.; Lee, J. H.; Jung, S. H.; Lee, K.; Lee, J. J. Bioorg. Med. Chem. Lett. 2007, 17, 6305-6310. https://doi.org/10.1016/j.bmcl.2007.09.005
  10. Won, M. S.; Im, N. H.; Park, S. H.; Boovanahalli, S. K.; Jin, Y. L.;Jin, X. J.; Chung, K. S.; Kang, M.; Lee, K.; Park, S. K.; Kim, H. M.;Kwon, B. M.; Lee, J. J.; Lee, K. Biochem. Biophys. Res. Commun.2009, 385, 16-21. https://doi.org/10.1016/j.bbrc.2009.05.022
  11. Lee, K.; Kang, J. E.; Park, S. K.; Jin, Y. L.; Chung, K. S.; Kim,H. M.; Lee, K.; Kang, M. R.; Lee, M. K.; Song, K. B.; Yang, E.G.; Lee, J. J.; Won, M. S. Biochem. Pharm. 2010, 80, 982-989. https://doi.org/10.1016/j.bcp.2010.06.018
  12. Maxwell, P. H.; Wiesener, M. S.; Chang, G.-W.; Clifford, S. C.;Vaux, E. C.; Cockman, M. E.; Wykoff, C. C.; Pugh, C. W.; Mather,E. R.; Ratcliffe, P. J. Nature 1999, 399, 271-275. https://doi.org/10.1038/20459

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  3. Recent advances in hypoxia-inducible factor (HIF)-1 inhibitors vol.49, pp.None, 2010, https://doi.org/10.1016/j.ejmech.2012.01.033
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