DOI QR코드

DOI QR Code

Synthesis of Bifunctional Chelating Agent Derived from Lysine and its Radiolabeling with 99mTc

  • Pyun, Mi-Sun (Radioisotope Research and Development Division, Nuclear Basic Science Department,Korea Atomic Energy Research Institute) ;
  • Choi, Kang-Hyuk (Radioisotope Research and Development Division, Nuclear Basic Science Department,Korea Atomic Energy Research Institute,) ;
  • Hong, Young-Don (Radioisotope Research and Development Division, Nuclear Basic Science Department,Korea Atomic Energy Research Institute) ;
  • Choi, Sun-Ju (Radioisotope Research and Development Division, Nuclear Basic Science Department,Korea Atomic Energy Research Institute)
  • Published : 2009.05.20

Abstract

Keywords

References

  1. Hung, M.; Huaang, Z. L.; Bilgen, M.; Berkland, C. Nanomedicine: Nanotechnology, Biology and Medicine, 2008, 4, 30 https://doi.org/10.1016/j.nano.2007.10.085
  2. Liu, S. Adv. Drug. Deliv. Rev. 2008, 60, 1347 https://doi.org/10.1016/j.addr.2008.04.006
  3. Yang, J. J.; Yang, J.; Wei, L.; Zurkiya, O.; Yang, W.; Li, S.; Zou, J.; Maniccia, A. L. W.; Mao, H.; Zhao, F.; Malchow, R.; Zhao, S.; Johnson, J.; Hu, Xiaoping.; Krogstad, E.; Liu, Z. R. J. Am. Chem. Soc. 2008, 130, 9260 https://doi.org/10.1021/ja800736h
  4. Yurt, A.; Kazanci, N. J. Mol. Struct. 2008, 892, 392 https://doi.org/10.1016/j.molstruc.2008.06.024
  5. Schibli, R.; Schubiger, P. A. Eur J. Nucl. Med. Mol. Imaging 2002, 29, 1529 https://doi.org/10.1007/s00259-002-0900-8
  6. Mundwiler, S.; Waibel, R.; Spingler, B.; Kunze, S.; Alberto, R. Nucl. Med. Biol. 2005, 32, 473 https://doi.org/10.1016/j.nucmedbio.2005.04.007
  7. Sunberg, M. W.; Meares, C. F.; Goodwin, D. A.; Diamanti, C. I. Nature 1974, 250, 587 https://doi.org/10.1038/250587a0
  8. Sundberg, M. W.; Meares, C. F.; Goodwin, D. A.; Diamanti, C. I. Med. Chem. 1974, 17, 1304 https://doi.org/10.1021/jm00258a015
  9. Chikara, B. S.; Kumar, N.; Tandon, V.; Mishra, A. K. Bioorgan. Med. Chem. 2005, 13, 4713 https://doi.org/10.1016/j.bmc.2005.04.073
  10. Schonherr, T.; Seichter, W.; Weber, E. Polyhedron 2006, 25, 3463 https://doi.org/10.1016/j.poly.2006.06.037
  11. Schonherr, T.; Weber, E.; Seichter, W. Z. Anorg. Allg. Chem. 2001, 627, 2420 https://doi.org/10.1002/1521-3749(200110)627:10<2420::AID-ZAAC2420>3.0.CO;2-X
  12. Miederer, M.; Scheinberg, D. A.; McDevitt, M. R. Adv. Drug. Deliv. Rev. 2008, 60, 1371 https://doi.org/10.1016/j.addr.2008.04.009
  13. Liang, X.; Parkinson, J. A.; Weishaupl, M.; Gould, R. O.; Paisey, S. J.; Park, H. S.; Hunter, T. M.; Blindauer, C. A.; Parsons, S.; Sadler, P. J. J. Am. Chem. Soc. 2002, 124, 9105 https://doi.org/10.1021/ja0260723
  14. Choi, K. H.; Hong, Y. D.; Pyun, M. S.; Choi, S. J. Bull. Korean Chem. Soc. 2006, 27, 1194 https://doi.org/10.5012/bkcs.2006.27.8.1194
  15. Arndt, F. Org. Synth. 1934, 2, 165
  16. Paquette, L. A. Encyclopedia of reagents for organic synthesis 1995, 2, 1512
  17. Martell, A. E.; Smith, R. M. Critical Stability Constants; Plenum Press: New York, 1974; p 204, p 236, p 281
  18. Zolle, I. Technetium-99m Pharmaceuticals Preparation and Quality Control in Nuclear Medicine; Springer: Berlin Heidelberg, New York, 2007; p 297-303

Cited by

  1. Preparation and preliminary biological evaluation of 177Lu-labeled GluDTPA-cyclo(RGDfK) for integrin ανβ3 receptor-positive tumor targeting vol.55, pp.1, 2011, https://doi.org/10.1002/jlcr.1944
  2. Dual modal imaging agents based on chromophore-bearing DTPA analogues vol.7, pp.61, 2017, https://doi.org/10.1039/C7RA06946D
  3. Effect of EDTA and PYP as Co-Ligand of Radiolabeled Nanomaterial M41S-NH2 for Radiosynovectomy vol.896, pp.1662-8985, 2014, https://doi.org/10.4028/www.scientific.net/AMR.896.687