DOI QR코드

DOI QR Code

An Efficient Synthesis of Racemic Tolterodine

  • Kang, Joo-Hi (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University) ;
  • Lee, Jong-Hyoup (Chirogenix Co., Ltd., Kowoon Institute of Technology Innovation, Suwon University) ;
  • Park, Young-Jun (Chirogenix Co., Ltd., Kowoon Institute of Technology Innovation, Suwon University) ;
  • Kim, Kyoung-Soo (Chirogenix Co., Ltd., Kowoon Institute of Technology Innovation, Suwon University) ;
  • Lee, Jae-Yeol (Research Institute for Basic Sciences and Department of Chemistry, College of Sciences, Kyung Hee University)
  • Published : 2008.02.20

Abstract

Keywords

References

  1. Jonas, U.; Hoefner, K.; Madersbacher, H.; Holmdahl, T. H. World J. Urol. 1997, 15, 144 https://doi.org/10.1007/BF02201987
  2. Gillberg, P. G.; Sundquist, S.; Nilvebrant, L. Eur. J. Pharmacol. 1998, 349, 285 https://doi.org/10.1016/S0014-2999(98)00214-3
  3. Yamanishi, T.; Chapple, C. R.; Chess-Williams, R. World J. Urol. 2001, 19, 299 https://doi.org/10.1007/s003450100226
  4. Sellers, D. J.; Yamanishi, T.; Chapple, C. R.; Couldwell, C.; Yasuda, K.; Chess-Williams, R. J. Auton. Pharmacol. 2000, 20, 171 https://doi.org/10.1046/j.1365-2680.2000.00181.x
  5. Hirose, H.; Aoki, I.; Kimura, T.; Fujikawa, T.; Numazawa, T.; Sasaki, K.; Nishikibe, M.; Noguchi, K. Eur. J. Pharmacol. 2002, 452, 245 https://doi.org/10.1016/S0014-2999(02)02335-X
  6. Nilvebrant, L.; Andersson, K. E.; Gillberg, P. G.; Stahl, M.; Sparf, B. Eur. J. Pharmacol. 1997, 327, 195 https://doi.org/10.1016/S0014-2999(97)89661-6
  7. Andersson, P. G.; Schink, H. E.; Osterlund, K. J. Org. Chem. 1998, 63, 8067 https://doi.org/10.1021/jo981259r
  8. Gage, J. R.; Cabaj, J. E. U.S. Patent 5,922,914, 1999
  9. Botteghi, C.; Corrias, T.; Marchetti, M.; Paganelli, S.; Piccolo, O. Org. Process Res. Dev. 2002, 6, 379 https://doi.org/10.1021/op020014k
  10. Selensky, C.; Pettus, T. R. R. J. Org. Chem. 2004, 69, 9196 https://doi.org/10.1021/jo048703c
  11. Colombo, L.; Rossi, R.; Castaldi, G.; Allegrini, P.; Dipharma, S. P. A. Italian Patent MI2004A000616, 2004; Canadian Patent CA 2502640, 2005; European Patent EP1584621, 2005
  12. Hedberg, C.; Andersson, P. G. Adv. Synth. Catal. 2005, 347, 662 https://doi.org/10.1002/adsc.200404234
  13. Chen, G.; Tokunaga, N.; Hayashi, T. Org. Lett. 2005, 7, 2285 https://doi.org/10.1021/ol0507367
  14. Ulgheri, F.; Marchetti, M.; Piccolo, O. J. Org. Chem. 2007, 72, 6056 https://doi.org/10.1021/jo0705667
  15. Srinivas, K.; Srinivasan, N.; Reddy, K. S.; Ramakrishna, M.; Reddy, C. R.; Arunagiri, M.; Kumari, R. L.; Venkataraman, S.; Mathad, V. T. Org. Process Res. Dev. 2005, 9, 314 https://doi.org/10.1021/op050024w
  16. Ulgheri, F.; Marchetti, M.; Piccolo, O. J. Org. Chem. 2007, 72, 6056 https://doi.org/10.1021/jo0705667
  17. Srinivas, K.; Srinivasan, N.; Reddy, K. S.; Ramakrishna, M.; Reddy, C. R.; Arunagiri, M.; Kumari, R. L.; Venkataraman, S.; Mathad, V. T. Org. Process Res. Dev. 2005, 9, 314 https://doi.org/10.1021/op050024w

Cited by

  1. ChemInform Abstract: An Efficient Synthesis of Racemic Tolterodine (VII). vol.39, pp.28, 2008, https://doi.org/10.1002/chin.200828095