References
- Radiotracer production. In: Wagner HN, Szabo Z, Buchanan JW, editiors. Principles of Nuclear Medicine Philadelphia: W.B. Saunders; 1995
- Snyder SE, Kilbourn MR. Chemistry of fluorine-18 radiopharmaceuticals. In: Welch MJ, Redvanly CS, editors. Handbook of Radiopharmaceuticals Chichester: Wiley; 2003. p 195-227
-
Pike VW, Eakins MN, Allan RM, Selwyn AP. Preparation of [
$1-^{11}C$ ]acetate - an agent for the study of myocardial metabolism by positron emission tomography. Int J Appl Radiat Isot 1982; 33:505-12 https://doi.org/10.1016/0020-708X(82)90003-5 -
Crouzel C, L
$\aa$ ngstr$\ddot{o}$ m B, Pike VW, Coenen HH. Recommendations for a practical production of [$^{11}$ C]methyl iodide. Appl Radiat Isot 1987;38:601-3 https://doi.org/10.1016/0883-2889(87)90123-7 -
Larsen P, Ulin J, Dahlström K, Jensen M. Synthesis of [
$^{11}$ C]iodomethane by iodination of [11C]methane. Appl Radiat Isot 1997;48:153-7 https://doi.org/10.1016/S0969-8043(96)00177-7 -
Jewett DM. A simple synthesis of [
$^{11}$ C]methyl triflate. Appl Radiat Isot 1992;43:1383-5 https://doi.org/10.1016/0883-2889(92)90012-4 -
N
$\aa$ gren K, Muller L, Halldin C, Swahn CG, Leuhkoinen P. Improved synthesis of some commonly used PET radioligands by the use of [$^{11}$ C]methyl triflate. Nucl Med Biol 1995;22:235-9 https://doi.org/10.1016/0969-8051(94)00083-V -
Comar D, Carton JC, Maziere M, Marazano C. labelling and metabolism of methionine-methyl-
$^{11}$ C. Eur J Nucl Med 1976; 1:11-4 - Iwata R, Pascali C, Bogni A, Miyake Y, Yanai K, Ido T. A simple loop method for the automated preparation of [11C]raclopride from [11C]methyl triflate. Appl Radiat Isot 2001;55:17-22 https://doi.org/10.1016/S0969-8043(00)00368-7
- Coenen HH. New radiohalogenation methods: An overview. In: Cox PH, Mather SJ, Sampson CB, Lazarus CR, editors. Progress in Radiopharmacy. Boston: Martinus Nijhoff; 1986. p 196-220
- Kim DW, Choe YS, Chi DY. A new nucleophilic fluorine-18 labeling method for aliphatic mesylates: reaction in ionic liquids shows tolerance for water. Nucl Med Biol 2003;30:345-50 https://doi.org/10.1016/S0969-8051(03)00017-9
-
Hamacher K, Coenen HH, Stöcklin G. Efficient stereospecific synthesis of no-carrier-added 2-[
$^{18}$ F]fluoro-2-deoxy-D-glucose using aminopolyether supported nucleophilic substitution. J Nucl Med 1986;27:235-8 -
Alauddin MM, Conti PS, Mazza SM, Hamzeh FM, Lever JR. 9-[(3-[
$^{18}$ F]-Fluoro-1-hydroxy-2-propoxy)methyl]guanine ([$^{18}$ F]-FHPG): a potential imaging agent of viral infection and gene therapy using PET. Nucl Med Biol 1996;23:787-92 https://doi.org/10.1016/0969-8051(96)00075-3 -
Haka MS, Kilbourn MR, Watkins GL, Toorongian SA. Aryltrimethylammonium trifluoromethanesulfonates as precursors to aryl [
$^{18}$ F]fluoride: Improved synthesis of [$^{18}$ F]GBR-13119. J Labelled Cpd Radiopharm 1989;27:823-33 https://doi.org/10.1002/jlcr.2580270711 -
Lee SY, Choe YS, Kim YR, Choi BW, Kim SE, Choi Y, Lee KH, Lee J, Kim BT. Synthesis and evaluation of
$^{18}$ F-labeled N-benzylpiperidine benzisoxazole for acetylcholinesterase mapping. J Nucl Med 2002;43S:358P -
Le Bars D, Lemaire C, Ginovart N, Plenevaux A, Aerts J, Brihaye C, et al. High-yield radiosynthesis and preliminary in vivo evaluation of p-[
$^{18}$ F]MPPF, a fluoro analog of WAY-100635. Nucl Med Biol 1998;25:343-50 https://doi.org/10.1016/S0969-8051(97)00229-1 -
Jonson SD, Welch MJ. Synthesis, biological evaluation, and baboon PET imaging of the potential adrenal agent cholesteryl-p-[
$^{18}$ F] fluorobenzoate. Nucl Med Biol 1999;26:131-8 https://doi.org/10.1016/S0969-8051(98)00081-X -
Ido T, Wan CN, Casella V, Fowler JS, Wolf AP, Reivich M, et al. Labeled 2-deoxy-2-fluoro-D-glucose analogs.
$^{18}$ F-Labeled 2-deoxy-2-fluoro-D-glucose, 2-deoxy-2-fluoro-D-mannose and$^{14}$ C-2-deoxy- 2-fluoro-D-glucose. J Labelled Cpd Radiopharm 1978;14:171-83 -
Fowler JS, Finn RD, Lambrecht RM, Wolf AP. The synthesis of
$^{18}$ F-5-fluorouracil. J Nucl Med 1973;14:63-4 -
Diksic M, Farrokhzad S, Yamamoto YL, Feindel W. A simple synthesis of
$^{18}$ F-labelled 5-fluorouracil using acetylhypofluorite. Int J Nucl Med Biol 1984;11:141-2 https://doi.org/10.1016/0047-0740(84)90049-4 -
Adam MJ, Jivan S. Synthesis and purification of L-6-[
$^{18}$ F] fluorodopa. Appl Radiat Isot 1988;39:1203-10 https://doi.org/10.1016/0883-2889(88)90100-1 - Hom RK, Katzenellenbogen JA. Technetium-99m-labeled receptorspecific small-molecule radiopharmaceuticals: recent developments and encouraging results. Nucl Med Biol 1997;24:485-98 https://doi.org/10.1016/S0969-8051(97)00066-8
- Jurisson SS, Lydon JD. Potential technetium small molecule radiopharmaceuticals. Chem Rev 1999;99:2205-18 https://doi.org/10.1021/cr980435t
- Spradau TW, Katzenellenbogen JA. Preparation of cyclopentadienyltricarbonylrhenium complexes using a double ligand transfer reaction. Organometallics 1998;17:2009-17 https://doi.org/10.1021/om971018u
-
Alberto R, Schibli R, Egli A, Schubiger AP. A novel organometallic aqua complex of technetium for the labeling of biomolecules: synthesis of [
$^{99m}Tc(OH_2)_3(CO)_3$ ]$^+$ - in aqueous solution and its reaction with a bifunctional ligand. J Am Chem Soc 1998;120:7987-8 https://doi.org/10.1021/ja980745t -
Kung MP. Stevenson DA, Pl
$\ddot{o}$ ssel K, Meegalla SK, Beckwith A, Essman WD, Mu M, Lucki I, Kung HF. [$^{99m}$ Tc]TRODAT-1: A novel technetium-99m complex as a dopamine transporter imaging agent. Eur J Nucl Med 1997;24:372-80 - Moerlein SM. Regiospecific aromatic radioiodination via n.c.a. copper (I) assisted iododebromination. Radiochim Acta 1990; 50:55-61
-
Neumeyer JL, Wang S, Milius RA. Baldwin RM, Zea-Ponce Y, Hofer PB, et al. [
$^{123}$ I]-2$\beta$ -Carbomethoxy-3$\beta$ -(4-iodophenyl)tropane: high-affinity SPECT radiotracer of monoamine reuptake sites in brain. J Med Chem 1991;34:3144-6 https://doi.org/10.1021/jm00114a027 -
Goodman MM, Kung M-P, Kabalka GW, Kung HF, Switzer R. Synthesis and characterization of radioiodinated N-(3-iodopropen-1-yl) 2
$\beta$ -carbomethoxy-3$\beta$ -(4-chlorophenyl)tropanes: potential dopamine reuptake site imaging agents. J Med Chem 1994;37:1535-42 https://doi.org/10.1021/jm00036a020 - Parker CW. Radiolabeling of proteins. Methods Enzymol 1990; 182:721-31 https://doi.org/10.1016/0076-6879(90)82056-8
- Blok D, Feitsma RIJ, Vermeij P, Pauwels EJK. Peptide radiopharmaceuticals in nuclear medicine. Eur J Nucl Med 1999; 26:1511-1519 https://doi.org/10.1007/s002590050488
- Fischman AJ, Babich JW. Radiolabeled paptides: a new class of imaging agents. In: Freeman LM, editor. Nuclear Medicine Annual. New York: Raven Press; 1997. p. 103
-
Wester H-J, Hamacher K, St
$\ddot{o}$ cklin G. A comparative study of N.C.A. fluorine-18 labeling of proteins via acylation and photochemical conjugation. Nucl Med Biol 1996;23:365-72 - King TP, Zhao SW, Lam T. Preparation of protein conjugates via intermolecular hydrazone linkage. Biochemistry 1986;25:5774-9 https://doi.org/10.1021/bi00367a064
- Rennen HJ, Boerman OC, Koenders EB, Oyen WJ, Corstens FH. Labeling proteins with Tc-99m via hydrazinonicotinamide (HYNIC): optimization of the conjugation reaction. Nucl Med Biol 2000; 27:599-604 https://doi.org/10.1016/S0969-8051(00)00134-7
-
Rennen HJ, Boerman OC, Oyen WJ, van der Meer JW, Corstens FH. Specific and rapid scintigraphic detection of infection with
$^{99m}$ Tc-labeled interleukin-8. J Nucl Med 2001;42:117-23 - Su Z-F, He J, Rusckowski M, Hnatowich. In vitro cell studies of technetium-99m labeled RGD-HYNIC peptide, a comparison of tricine and EDDA as co-ligands. Nucl Med Biol 2003;30:141-9 https://doi.org/10.1016/S0969-8051(02)00390-6
- Russell J, O'Donoghue JA, Finn R, Koziorowski J, Ruan S, Humm JL, et al. Iodination of annexin V for imaging apoptosis. J Nucl Med 2002;43:671-7
- Bolton AM, Hunter RM. The labeling of proteins to high specific radioactivities by conjugation to I-125 containing acylating agent. Biochem J 1973;133:529-39 https://doi.org/10.1042/bj1330529
- Zalutsky MR, Narula AS. A method for the radiohalogenation of proteins resulting in decreased thyroid uptake of radioiodine. Appl Radiat Isot 1987;38:1051-5 https://doi.org/10.1016/0883-2889(87)90069-4