참고문헌
- Neu, H. C. : The crisis in antibiotic resistance. Science 257, 1064 (1992) https://doi.org/10.1126/science.257.5073.1064
-
Reading,C. and Cole, M. : Clavulanic acid : A
${\beta}$ lactamaseinhibiting${\beta}$ lactam from Streptomyces clavuligerus. Antimicrob.Agents Chemother. 11, 852 (1977) -
English, A. R., Retsema, J. A., Girard, A. E., Lynch, J. E. and Barth, W. E. : CP-45,899, a
${\beta}$ -lactamase inhibitor that extends the antibacterial spectrum of${\beta}$ -lactams; initial bacteriological characterization. Antimicrob. Agents. Chemother 14, 414 (1978) -
Micetich, R. G., Maiti, S. N., Spevak, P., Hall, T. W., Yamabe, S., Ishida, N., Tanaca, M., Yamazaki, T., Nakai, A. and Ogawa, K. : Synthesis and
${\beta}$ -lactamase inhibitory properties of 2${\beta}$ -[(1,2,3-triazol-1-yl)methyl]-2${\alpha}$ -methylpenam-3${\alpha}$ -carboxylic acid 1,1-dioxide and related triazolyl derivatives. J. Med. Chem. 30, 1469 (1987). https://doi.org/10.1021/jm00391a032 -
Chen, Y. L., Chang, C. W. and Hedberg, K. : Synthesis of a potent
${\beta}$ -lactamase inhibitor 1, 1-dioxo-6-(2-pyricyl)methyl enepenicillanic acid and its reaction with sodium methoxide. Tetrahedron Lett. 27, 3449 (1986) https://doi.org/10.1016/S0040-4039(00)84819-4 -
Bennett, I. S., Brooks, G., Broom, N. J., Calvert, S. H., Coleman, K. and Francois, I. : 6-(Substituted methylene) penems, potent broad spectrum inhibitors of bacterial
${\beta}$ -lactamase V. Chiral 1,2,3-triazolyl derivatives. J. Aniibiotics 44, 969 (1991) -
Bennett , I., Broom, N. J., Bruton, G., Calvert, S., Clarke, B. P., Coleman, K., Edmondson, R., Edwards, P., Jones, D., Osborne, N. F. and Walker, G. : 6-(Substituted methyler.e)penems, potent broad spectrum inhibitors of bacterial -
${\beta}$ lactamase III. Structure-activity relationships of the 5-membered heterocyclic derivatives. J. Antibiotics 44, 331 (1991) -
Broom, N. J. P., Brooks, G. and Clark, B. P. :
${\beta}$ -(Substituted methylene) penems. Eur. Pat. Appl. 321187 AI, (1989) -
Chen, Y. L., Chang, C. w., Hedberg, K., Guarino,K., Welch, W. M. and Kiessling, L. : Structure-activity relatiomships of 6(heterocyclyl) methylene penam sulfones; a new class of
${\beta}$ -lactamase inhibitors. J. Antibiotics 40, 803 (1987) - Boyer, J. H. and Hamer, J. : The acid-catalyzedreaction of alkyl azides upon carbonyl compounds. J. Am. Chem. Soc. 77, 951 (1995) https://doi.org/10.1021/ja01609a045
- Sauer, J. C. : In Organic syntheses Collective volume IV., Robjohn, John Wiley and Sons, Inc., New York, 813 (1963)