DOI QR코드

DOI QR Code

Protein Tyrosine Phosphatase 1B Inhibitors: Catechols

  • Ahn, Jin-Hee (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Cho, Sung-Yun (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Ha, Jae-Du (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Kang, Seung-Kyu (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Jung, Sun-Ho (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Kim, Hye-Min (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Kim, Sung-Soo (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Kim, Kwang-Rok (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Cheon, Hyae-Gyeong (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Yang, Sung-Don (Medicinal Science Division, Korea Research Institute of Chemical Technology) ;
  • Choi, Joong-Kwon (Medicinal Science Division, Korea Research Institute of Chemical Technology)
  • Published : 2003.10.20

Abstract

Keywords

References

  1. Saltiel, A. R.; Kahn, C. R. Nature 2001, 414, 799. https://doi.org/10.1038/414799a
  2. Elchebly, M.; Payette, P.; Michaliszyn, E.; Cromlish, W.; Collins, S.; Loy, A. L.; Normandin, D.; Cheng, A.; Himms-Hagen, J.;Chan, C.-C.; Ramachandran, C.; Gresser, M. J.; Tremblay, M. L.;Kennedy, B. P. Science 1999, 283, 1544. https://doi.org/10.1126/science.283.5407.1544
  3. Johnson, T. O.; Ermolieff, J.; Jirousek, M. R. Nature Reviews/Drug Discovery 2002, 1, 696. https://doi.org/10.1038/nrd895
  4. van Huijsduijnen, R. H.; Bombrun, A.; Swinnen, D. DrugDiscovery Today 2002, 7, 1013. https://doi.org/10.1016/S1359-6446(02)02438-8
  5. Ahn, J. H.; Cho, S. Y.; Ha, J. D.; Chu, S. Y.; Jung, S. H.; Jung,Y. S.; Baek, J. Y.; Choi, I. K.; Shin, E. Y.; Kang, S. K.; Kim, S. S.;Cheon, H. G.; Yang, S. D.; Choi, J.-K. Bioorg. Med. Chem. Lett.2002, 12, 1941. https://doi.org/10.1016/S0960-894X(02)00331-1
  6. Cho, S. Y.; Ahn, J. H.; Ha, J. D.; Kang, S. K.;Jung, S. H.; Kim, H.-M.; Baek, J. Y.; Han, S. S.; Shin, E. Y.; Kim,S. S.; Kim, K. R.; Cheon, H. G.; Yang, S. D.; Choi, J.-K. Bull.Korean Chem. Soc. 2003, in press.
  7. Kumar, P. Org. Prep. Proceed. Inter. 1997, 29, 477. https://doi.org/10.1080/00304949709355222
  8. Christoffers, J.; Mann, A. Eur. J. Org. Chem. 2000, 1977.
  9. Itoh, S.; Fukui, Y.; Haranou, S.; Ogino, M.; Komatsu, M.;Ohshiro, Y. J. Org. Chem. 1992, 57, 4452. https://doi.org/10.1021/jo00042a028

Cited by

  1. Synthesis of (±)-Brazilin Using IBX vol.7, pp.26, 2005, https://doi.org/10.1021/ol0523749
  2. Dual colorimetric and fluorogenic probes for visualizing tyrosine phosphatase activity vol.53, pp.14, 2017, https://doi.org/10.1039/C6CC09204G
  3. Protein Tyrosine Phosphatase 1B Inhibitors: A Molecular Level Legitimate Approach for the Management of Diabetes Mellitus vol.32, pp.3, 2012, https://doi.org/10.1002/med.20219
  4. Protein Tyrosine Phosphatase 1B Inhibitors: Catechols. vol.35, pp.8, 2003, https://doi.org/10.1002/chin.200408100
  5. A Facile Synthesis of Cyclopenta[d][1,2]oxazines through [6+4] Cycloaddition Reaction vol.27, pp.9, 2003, https://doi.org/10.5012/bkcs.2006.27.9.1481
  6. Privileged Structure-based Discovery of Novel 2-Iminothiazoles as Protein Tyrosine Phosphatase 1B Inhibitors vol.34, pp.10, 2003, https://doi.org/10.5012/bkcs.2013.34.10.2861