Bulletin of the Korean Chemical Society

Korean Chemical Society (대한화학회)
권호 표지
DOI QR코드

DOI QR Code

Synthesis of Novel Quinolinecarboxamide Derivatives with Estrogenic Activity

  • Um, Soo-Jong (Dept. of Bioscience & Biotechnology/Institute of Bioscience, Sejong University) ;
  • Park, Si-Ho (Chebigen Inc., 305-B, Chungmugwan, Sejong University) ;
  • Park, Chong-Ho (Dept. of Bioscience & Biotechnology/Institute of Bioscience, Sejong University) ;
  • Chang, Byung-Ha (IDR Tech., Inc., Research center B-1, Kwacheon Officetel 5th Fl.) ;
  • Yoon, Jeong-Hyeok (IDR Tech., Inc., Research center B-1, Kwacheon Officetel 5th Fl.) ;
  • Sin, Hong-Sig (Chebigen Inc., 305-B, Chungmugwan, Sejong University)
  • Published : 2003.05.20
Download PDF
⟨ Previous Next ⟩

Abstract

Keywords

References

  1. Dickinson, R. B.; McManaway, M. E.; Lippman, M. E. Science1986, 232, 1540. https://doi.org/10.1126/science.3715461
  2. Tsai, M. J.; OMalley, B. W. Annul. Rev. Biochem. 1994, 63, 451. https://doi.org/10.1146/annurev.bi.63.070194.002315
  3. Sun, J.; Meyers, M. J.; Fink, B. E.; Rajendran, R.; Katzenellenbogen,J. A.; Katzenellenbogen, B. S. Endocrinology 1999, 140, 800. https://doi.org/10.1210/en.140.2.800
  4. Wiese, T. E.; Polin, L. A.; Palomino, E.; Brooks, S. C. J. Med.Chem. 1997, 40, 3659. https://doi.org/10.1021/jm9703294
  5. Li, J. J.; Hou, X.; Bentel, J.; Yazlovitskaya, E. M.; Li, S. A.Carcinogenesis 1998, 19, 471. https://doi.org/10.1093/carcin/19.3.471
  6. Lippman, M. E.; Bolan, G. Nature 1975, 256, 592. https://doi.org/10.1038/256592a0
  7. Jordan, V. C. Eur. J. Cancer 1976, 12, 419. https://doi.org/10.1016/0014-2964(76)90030-X
  8. Jordan, V. C.; Morrow, M. Br. Med. J. 1999, 319, 331. https://doi.org/10.1136/bmj.319.7206.331
  9. Munster, P. N.; Buzdar, A.; Dhingra, K.; Enas, N.; Ni, L.; Major,M.; Melemed, A.; Seidman, A.; Booser, D.; Theriault, R.; Norton,L.; Hudis, C. J. Clin. Oncol. 2001, 19, 2002.
  10. Labrie, F.; Labrie, C.; Belanger, A.; Simard, J.; Gauthier, S.; Luu-The, V.; Merand, Y.; Giguere, V.; Candas, B.; Luo, S.; Martel, C.;Singh, S. M.; Fournier, M.; Coquet, A.; Richard, V.; Charbonneau,R.; Charpenet, G.; Tremblay, A.; Tremblay, G.; Cusan, L.;Veilleux, R. J. Steroid Biochem. Mol. Biol. 1999, 69, 51. https://doi.org/10.1016/S0960-0760(99)00065-5
  11. Ke, H. Z.; Qi, H.; Chidsey-Frink, K. L.; Crawford, D. T.;Thompson, D. D. J. Bone Miner. Res. 2001, 16, 765. https://doi.org/10.1359/jbmr.2001.16.4.765
  12. Doebner, O. Ber. 1883, 16, 2357. https://doi.org/10.1002/cber.188301602155
  13. Atwell, G. J.; Baguley, B. C.; Denny, W. A. J. Med. Chem. 1989,32, 396. https://doi.org/10.1021/jm00122a018
  14. Dhaon, M. K.; Olsen, R. K.; Ramasamy, K. J. Org. Chem.1982, 47, 1962. https://doi.org/10.1021/jo00349a028
  15. Desai, M. C.; Stephens Stramiello, L. M.Tetrahedron Lett. 1993, 34, 7685. https://doi.org/10.1016/S0040-4039(00)61539-3
  16. Akaji, K.; Kuriyama, N.; Kiso, Y. Tetrahedron Lett. 1994, 35, 3315. https://doi.org/10.1016/S0040-4039(00)76895-X
  17. Norman, B. H.; Hemscheidt, T.; Schultz, R. M.; Andis, S. L. J. Org. Chem. 1998, 63, 5288. https://doi.org/10.1021/jo980536r
  18. Saari, W. S.; Schwering, J. E.; Lyle, P. A.; Smith, S. J.; Engelhardt,E. L. J. Med. Chem. 1990, 33, 97. https://doi.org/10.1021/jm00163a016
  19. Fletcher, S. R.; Burkamp, F.; Blurton, P.; Cheng, S. K. F.;Clarkson, R.; O'Connor, D.; Spinks, D.; Tudge, M.; van Niel, M.B.; Patel, S.; Chapman, K.; Marwood, R.; Shepheard, S.; Bentley,G.; Cook, G. P.; Bristoww, L. J.; Castro, J. L.; Hutson, P. H.;MacLeod, A. M. J. Med. Chem. 2002, 45, 492. https://doi.org/10.1021/jm011030v
  20. Salvatore, R. N.; Yoon, C. H.; Jung, K. W. Tetrahedron 2001, 57, 7785. https://doi.org/10.1016/S0040-4020(01)00722-0
  21. Um, S. J.; Kim, E. J.; Hwang, E. S.; Kim, S. J.; Namkoong, S. E.; Park, J. S. Int. J. Cancer 2000, 85, 416. https://doi.org/10.1002/(SICI)1097-0215(20000201)85:3<416::AID-IJC19>3.0.CO;2-3

Cited by

  1. Design, synthesis, and cytotoxic activities of new 2,4,5-triarylimidazoles vol.22, pp.8, 2013, https://doi.org/10.1007/s00044-012-0391-5
  2. Synthesis of Novel Quinolinecarboxamide Derivatives with Estrogenic Activity. vol.34, pp.43, 2003, https://doi.org/10.1002/chin.200343126
  3. Multicomponent cyclocondensation reactions of aminoazoles, arylpyruvic acids and aldehydes with controlled chemoselectivity vol.64, pp.49, 2003, https://doi.org/10.1016/j.tet.2008.09.089
  4. Heterocyclization Reactions of Pyruvic Acids and Aminoazoles with Controlled Chemoselectivity vol.3, pp.2, 2003, https://doi.org/10.17721/fujcv3i2p1-20