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Synthesis of Pyrazinopsoralen : A Pyrazine Ring Fused Monofunctional Psoralen Derivative

  • 발행 : 1995.12.20

초록

An efficient synthesis of 6,8-dioxa-1,4-diazacyclopenta[b]phenanthren-5-one (Pyrazinopsoralen) (4) has been carried out by the Suzuki coupling reaction as a key step starting from 5-bromo-6-methoxybenzofuran (6) and methyl 2-iodo-3-pyrazinecarboxylate (8).

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참고문헌

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