Synthesis of New Benzimidazo [2,1-b][1,3,5]benzothiadiazepine Derivatives

새로운 Benzimidazo[2,1-b][1,3,5]benzothiadiazepine 유도체들의 합성

  • 진병우 (중앙대학교 이과대학 화학과) ;
  • 조성희 (중앙대학교 화학과)
  • Published : 19940500

Abstract

New 6-imino-5H-benzimidazo[2,1-b][1,3,5]benzothiadiazepine derivatives (8) were successfully synthesized in good yields from the N-[2-(benzimidazol-2-yl thio)phenyl]thiourea derivatives (6) in the presence of dicyclohexylcarbodiimide(DCC) and from N-[2-(benzimidazol-2-yl thio)phenyl]-S-methylisothiourea derivatives (7) with potassium carbonate.

새로운 6-imino-5H-benzimidazo[2,1-b][1,3,5]benzothiadiazepine 유도체(8)들을 dicyclohexylcarbodiimide(DCC)를 사용하여 N-[2-(benzimidazol-2-yl thio)phenyl]thiourea 유도체(6)로부터 합성하거나 potassium carbonate를 사용하여 N-[2-(benzimidazol-2-yl thio)phenyl]thiourea 유도체(7)로 부터 합성하였다.

Keywords

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