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Synthesis of 1-(N-carbobenzoxythiazolidinyl)-2-hydroxy-3-ethoxycarbonyl-1,2,3,4-tetrahydro-${\beta}$-carboline

  • Byung Hee Yoon (Department of Chemistry, Yonsei University) ;
  • Hak Soo Lyu (Department of Chemistry, Yonsei University) ;
  • Jee Hyun Hahn (Department of Chemistry, Yonsei University) ;
  • Chan Mug Ahn (Department of Chemistry, Yonsei University Wonju College of Medicine)
  • Published : 1991.08.20

Abstract

Pictet-Spengler reaction of the N-hydroxytryptophan ethyl ester (4) with N-protected thiazolidine aldehyde (8) has been carried out. The product, compound (9b), might be a possible precursor for the eudistomins C, E, K, and L.

Keywords

References

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