Synthesis and Anti-Inflammatory and Analgesic Activities of 2,4-Di-n-butyl-3,5-diarylimino-1,2,4-thiadiazolidines

  • Pandeya, S.N. (Department of Pharmaceutics, Institute of Technology) ;
  • Naik, P.R. (Banaras Hindu University) ;
  • Singh, S. (Banaras Hindu University) ;
  • Singh, P.N. (Banaras Hindu University)
  • Published : 1991.03.01

Abstract

Ten 1,2,4-thiadiazolidines were synthesized and screened for their anti-inflammatory and analgesic activities. Butyl isothiocyanate was used as a starting material. Several compounds showed significant anti-inflammatory and analgesic activities. The unsubstituted and o-methyl, p-acetoxy and o-chloro substituted compounds were found to be more potent anti-inflammatory and analgesic agents than the other compounds.

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